Three-Component Synthesis of Polysubstituted Homoproline Analogs
نویسندگان
چکیده
منابع مشابه
Three-component synthesis of polysubstituted homoproline analogs.
Tetrasubstituted pyrrolidines representing analogs of homoproline were synthesized by three-component condensation of aryl(heteroaryl)aldehydes, asparagine and N-methylmaleimide (NMM). Compounds with (1S*, 3R*, 3aS*, 6aR*)-configuration at the corresponding carbon positions of the bicyclic pyrrolidine ring could be isolated ona preparative scale.
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ژورنال
عنوان ژورنال: Molecules
سال: 2005
ISSN: 1420-3049
DOI: 10.3390/10070755